Hormonal Regulation

Argipressin

Also known as: AVP, Vasopressina, ADH

Molecular Identifiers

Molecular Formula

C46H65N15O12S2

PubChem CID

644077

Molecular Weight

1084.23 Da

Overview

Cyclic antidiuretic hormone (ADH) with a disulfide bridge. Produced in the hypothalamus and released by the neurohypophysis. Regulates water reabsorption in the kidneys, vasoconstriction, and body fluid homeostasis.

Sequence (1 letter): CYFQNCPRG
Extended notation: Cys-Tyr-Phe-Gln-Asn-Cys-Pro-Arg-Gly

Half-life

~10-20 minutes

Administration Route

Intravenous or subcutaneous

Category

Hormonal Regulation

Mechanism of Action

  • V1a receptor agonism (vasoconstriction)
  • V2 receptor agonism (water reabsorption in renal collecting ducts)
  • V1b receptor agonism (ACTH release from the pituitary)
  • Aquaporin-2 insertion into the apical membrane of collecting ducts
  • Regulation of plasma osmolality and blood volume

Dosage Protocol

Data compiled from the literature. This does not constitute medical advice.

Parameter Value
Dose 5-20 IU or 1-4 mcg/kg
Frequency As clinically needed
Timing Per protocol
Duration As needed

Reported Side Effects

Adverse effects described in the literature. Severity and frequency vary between individuals.

  • Nausea
  • Abdominal cramps
  • Pallor
  • Transient hypertension
  • Bradycardia

Presentations & Preparation

Vials of Argipressin found in the research market:

5 mg10 mg

Reconstitution

  • Diluent: Bacteriostatic water
  • Volume: 1 ml per vial
  • Inject the diluent slowly against the vial wall
  • Gently swirl until fully dissolved
  • Never shake

Storage

  • Lyophilized: Refrigerated 2-8°C
  • Reconstituted: Refrigerated 2-8°C (use within 24 hours)
  • Protect from direct light
  • Sensitive to degradation - use promptly after reconstitution
Reconstitution Calculator

Related Peptides