GH Secretagogues

MK-677

Also known as: Ibutamoren, MK-0677, L-163,191

Molecular Identifiers

Molecular Formula

C27H36N4O5S

CAS Number

159752-10-0

PubChem CID

6450830

Molecular Weight

528.67 Da

Overview

Oral non-peptidic ghrelin receptor (GHS-R1a) agonist that promotes sustained GH and IGF-1 secretion. Unlike GHRP peptides, it is orally bioavailable with a long half-life, maintaining elevated GH levels for up to 24 hours.

Small non-peptidic molecule. Oral ghrelin receptor agonist.

Half-life

~24 hours

Administration Route

Oral

Category

GH Secretagogues

Mechanism of Action

  • Oral ghrelin receptor (GHS-R1a) agonism
  • Sustained GH secretion for 24 hours
  • Elevation of serum IGF-1
  • Mimicry of physiological GH pattern (amplified pulses)
  • Appetite increase via ghrelin signaling

Dosage Protocol

Data compiled from the literature. This does not constitute medical advice.

Parameter Value
Dose 10-25 mg per dose
Frequency Once daily
Timing Before bedtime (to minimize GH effects on sleep)
Duration 8-12 weeks

Reported Side Effects

Adverse effects described in the literature. Severity and frequency vary between individuals.

  • Increased appetite (very common)
  • Water retention
  • Numbness/tingling
  • Elevated blood glucose
  • Lethargy
  • Joint pain

Product Properties

Purity >99%
Appearance White capsules or tablets
Source Chemical synthesis

Presentations & Preparation

Vials of MK-677 found in the research market:

10 mg (60 cápsulas)25 mg (60 cápsulas)

Reconstitution

  • Diluent: N/A (capsules or tablets)
  • Volume: N/A
  • Supplied as capsules or tablets
  • Administer with or without food

Storage

  • Lyophilized: Room temperature
  • Reconstituted: N/A
  • Keep in a dry place
  • Protect from light and moisture
Reconstitution Calculator

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