Cognitive & Neuroprotective

DSIP

Also known as: Peptídeo Indutor de Sono Delta

Molecular Identifiers

Molecular Formula

C35H48N10O15

CAS Number

62568-57-4

PubChem CID

68816

Molecular Weight

848.8 Da

Overview

Neuropeptide that regulates sleep and circadian rhythms. Induces delta wave sleep (deep sleep) without forced sedative effect. Acts on neuroendocrine modulation and possesses adaptogenic and antioxidant properties.

The interest in DSIP lies in the regulation of deep sleep: it induces the delta wave phase without the forced sedative effect typical of classical hypnotics, modulates circadian rhythms, and has adaptogenic and antioxidant properties. It is proposed in chronic insomnia, adrenergic stress, and as support for physical recovery, with effects also on neuroendocrine regulation (ACTH, cortisol, LH).

It has no approval as a medicine by the FDA, EMA, or ANVISA. In the peptide market it circulates through compounding pharmacies and specialized suppliers, in short cycles of 2-4 weeks, with subcutaneous administration 30-60 minutes before bedtime. The half-life is very short (~15-25 minutes), so the clinical effect appears to result from a signaling cascade rather than the sustained presence of the peptide.

It was characterized in the 1970s from research on rabbit blood during the delta phase of sleep, led by the Schoenenberger and Monnier group in Switzerland. Clinical evidence in humans is old and scarce, with most publications concentrated in the 1980s-90s.

Sequence (1 letter): WAGGDASGE
Extended notation: Trp-Ala-Gly-Gly-Asp-Ala-Ser-Gly-Glu

Half-life

~15-25 minutes

Administration Route

Subcutaneous or intravenous

Category

Cognitive & Neuroprotective

Mechanism of Action

  • Induction of delta wave sleep (restorative deep sleep)
  • Modulation of circadian rhythms and the sleep-wake cycle
  • Neuroendocrine regulation (ACTH, cortisol, LH)
  • Antioxidant and anti-stress properties
  • Limitation of oxidative stress at the cellular level

Dosage Protocol

Data compiled from the literature. This does not constitute medical advice.

Parameter Value
Dose 100-300 mcg per subcutaneous injection
Frequency Once daily
Timing 30-60 minutes before bedtime
Duration 2-4 weeks

Reported Side Effects

Adverse effects described in the literature. Severity and frequency vary between individuals.

  • Daytime drowsiness
  • Mild morning headache
  • Dizziness

Product Properties

Purity >98%
Appearance White lyophilized powder
Solubility Soluble in water and bacteriostatic water
Source Solid-phase peptide synthesis (SPPS)
Storage Lyophilized: -20°C for up to 2 years, 2-8°C for up to 6 months. Reconstituted: 2-8°C for up to 4 weeks. Protect from light and moisture. Avoid repeated freeze-thaw cycles.

Presentations & Preparation

Vials of DSIP found in the research market:

5 mg10 mg15 mg20 mg

Reconstitution

  • Diluent: Bacteriostatic water
  • Volume: 2 ml per vial
  • Inject the diluent slowly against the vial wall
  • Gently swirl until fully dissolved
  • Never shake

Storage

  • Lyophilized: Refrigerated 2-8°C
  • Reconstituted: Refrigerated 2-8°C (up to 30 days)
  • Protect from direct light
  • Do not freeze after reconstitution
Reconstitution Calculator

Scientific Studies

Published studies on DSIP.

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